Welcome to Astor Scientific

New collections added! Learn more

Popular right now
Lots of people have looked at this recently

Selling fast!
Grab yours while you can

TribioScience | SKU: TBI4814-10MG

Linsitinib, IGF-1R kinase and InsR kinase inhibitor (TBI4814)

Name: Linsitinib, IGF-1R kinase and InsR kinase inhibitor (TBI4814)
Brand: TribioScience
SKU: TBI4814-10MG
Price: 108.0 USD
Availability: InStock

$108.00

Shipping calculated at checkout.

Option

Product variants

Care information

Display general product information or specific product information using metafields.

Delivery and Shipping

Add some general information about your delivery and shipping policies.

Payment & Security

Payment methods

Your payment information is processed securely. We do not store credit card details nor have access to your credit card information.

Product Description

Product Reviews

TribioScience

Linsitinib, IGF-1R kinase and InsR kinase inhibitor (TBI4814)

From $108.00

Description

Product Details

Formal Name: 3-[8-Amino-1-(2-phenyl-7-quinolyl)imidazo[1,5-a]pyrazin-3-yl]-1-methyl-cyclobutanol

Alternate Names: OSI-906

Molecular Formula: C₂₆H₂₃N₅O

Formula Weight: 421.49

CAS Number: 867160-71-2

Purity: >98%

Formulation: powder

Solubility: Soluble in DMSO (up to 30 mg/ml).

Storage: -20°C

Stability: ≥ 1 year.

Applications

IGF-1R kinase and InsR kinase inhibitor

Functions

Linsitinib is a potent and selective dual inhibitor of insulin-like growth factor 1 (IGF-1R) kinase and insulin receptor (InsR) kinase (IC50’s = 35 and 75 nM respectively). It has been investigated as a chemotherapeutic in combination with other drugs for various cancers.