CL-82198, MMP-13 inhibitor (TBI1028)

Description

Product Details

Formal Name: N-[4-(4-Morpholinyl)butyl]-2-benzofurancarboxamide

Molecular Formula: C₁₇H₂₂N₂O₃

Formula Weight: 302.37

CAS Number: 307002-71-7

Purity: >98%

Formulation: powder

Solubility: Soluble in DMSO (up to 10 mg/ml).

Storage: RT

Stability: ≥ 2 years.

Applications

MMP-13 inhibitor

Functions

Selective inhibitor of MMP-13 (IC50 = 10 µM). It displayed no activity against MMP-1, MMP-9 or TACE.

Application Procedures

First dissolved in DMSO (up to 10 mg/ml), then diluted to aqueous buffer. Solutions in DMSO may be stored at -20°C for up to 6 months.